Kuunzwa kweCitrus Aurantium Extract

Kuunzwa kweCitrus Aurantium

Citrus Aurantium, chirimwa chemhuri yerutaceae, chinopararira zvakanyanya muChina. Citrus aurantium izita rechiChinese rekuti lime. Mukurapa kwechivanhu kwechiChinese, citrus aurantium imuriwo wechivanhu unoshandiswa zvakanyanya kuwedzera chido chekudya uye kudzora qi (simba). MuItaly, citrus aurantium yave iriwo mushonga wechivanhu kubvira muzana remakore rechi16, uchishandiswa kurapa fivha yakaita semarariya uye semushonga unorwisa utachiona. Ongororo dzichangobva kuitwa dzakaratidza kuti citrus aurantium inogona kutsiva ephedra mukurapa kufuta pasina migumisiro yakaipa yemwoyo.

Chinhu chinoshanda che citrus aurantium ndihesperidin, neohesperidin, nobiletin, auranetin, aurantiamarin, nuringin, synephrine, limonin.

Citrus Aurantium Extract-Ruiwo

 

Chinhu chinoshanda

hesperidin, neohesperidin, nobiletin, D-limonene, auranetin, aurantiamarin, citrin, synephrine, limonin

Zvivakwa zvemuviri

Kugayiwa kwekristaro, pokunyunguduka 184-1850C, kugayiwa kwekristaro kabhoni 151-152, kunonyunguduka nyore mumvura. Bitartrate, pokunyunguduka 188-189, kunonyunguduka mumvura, kunonetsa kunyunguduka muethanol, kunoda kusanyunguduka muchloroform, ether. Hydrochloride, kristaro isina ruvara (ethanol-ethyl ether), pokunyunguduka 166-167. Kugayiwa kwekristaro kuri nyore kuitika mukupatsanurwa kwechromatography kwe strong acid uye base ion exchange resins.

Mhedzisiro yemishonga
1. Mhedzisiro pachibereko: Fructus Aurantii naFructus Aurantii Fructus Decoction kubva munzvimbo nhatu dzakasiyana dzinobereka (Sichuan, Jiangxi, naHunan) yakaratidza mhedzisiro yekudzivirira chibereko mu vitro yemakonzo (ane pamuviri neasina pamuviri); Chibereko chetsuro chakafara mu vitro uye mu vitro (ane pamuviri uye asina pamuviri). Fistula yechibereko chetsuro yakaratidzawo kuti chiuno chechibereko chakasimba, kuwedzera kushushikana, uye kunyange tetanic contraction. Fructus Aurantii tincture uye Fructus Aurantii fluid extract zvinogonawo kumutsa chibereko chetsuro (mu vitro uye mu vitro). Chibereko chemumbeva (mu vitro) chakadziviswa. Chinhu chealkaloid chakabviswa kubva kuFructus Aurantii naLycium orange chaivewo nemhedzisiro yakati yekubata chibereko chetsuro mu vitro, kunyanya pamhasuru yechibereko yakamutswa nepituitrin. Chikamu chealkaloid chakabviswa chaive nemhedzisiro yekuzorora pachibereko chetsuro mu vitro, uye mhedzisiro yekuzorora yechibereko yaive pachena mushure mekusagadzikana kwemuviri. Cirantin, yakabviswa kubva kuFructus Aurantii Fructus Peel, inodzivirira hyaluronate yakakomberedza ovary, izvo zvingave zvine chekuita nemhedzisiro yayo yekudzivirira pamuviri (kudzivirira kubereka).

2. Mhedzisiro paura: Fructus Aurantii naFructus Aurantii vanobva munzvimbo nhatu dzakasiyana vakadzivisa ura mumakonzo netsuro; Matubhu mazhinji emudumbu mutsuro akadziviswa, asi mashoma haana kuchinja. Fructus Aurantii nemvura yainobva mudumbu yakadzivisa matubhu emudumbu emakonzo (in vitro) netsuro (in vitro). Kuwanda kwakanyanya (1:1000) kwakadzivisa ura hudiki hwetsuro dzakaparadzana nenguruve dzemuGuinea uye kwakadzivisa migumisiro yeacetylcholine nehistamine. Kuwanda kwakaderera (1:10 000), mushure menguva pfupi yekudziviswa, kunogona kuratidza mhedzisiro yekumutsa, amplitude yakawedzera, uye frequency yakawedzera. Mumbwa dzakarapwa, kuvapo kweura kwakadziviswa zviri pachena ne decoctions. Asi kune imbwa dzine gastroenterostomy, ine imwe mhedzisiro yekumutsa, iyo inogona kuita kuti kufamba kwemudumbu uye contraction rhythm ive nesimba.

3. Mhedzisiro pamwoyo netsinga dzeropa: kushoma kwekufara uye kudzikisira kukuru pamoyo wegudo in vitro. Fructus Aurantii naFructus Aurantii Aurantii decoction yemvura, Fructus Aurantii tincture, uye fluid extract zvakafanana. Fructus Aurantii decoction kana alcohol extract inopinzwa mutsinga inogona kukonzera kuwedzera kukuru kwekumanikidza. Fructus Aurantii naFructus Aurantii Fructus inobva munzvimbo nhatu dzakasiyana yakaratidzwa kuti ine mhedzisiro yekudzikisa kusimba kweropa nekubuda kweropa kwegudo mumuviri wese. Mumbwa dzakarapwa, paive nemhedzisiro yakakosha uye inokurumidza yeBP. Pakanga pasina kuora mwoyo kwekufema kana hypotension yakakonzerwa ne epinephrine, uye pakanga pasina kuwedzera kuri pachena kwekurova kwemoyo.

Maitiro ekuwedzera kumanikidzwa ane chekuita nezvinhu zvinotevera:

3.1. Kufadzwa kweα receptors, zvichikonzera kuvharika kweropa mumimwe mitezo yemuviri (phenylzoline inogona kudzosera simba rekuwedzera kweropa kuita kuti ropa ridzikire).

3.2. Kuwedzerwa kwemwoyo uye kuwedzera kwesimba remwoyo (kuyerera kweropa mumoyo wenguruve yegaini uye kugadzirira kwemoyo nemapapu). Mushure me reserpine, simba reFructus aurantii aurantii raiwedzera kumanikidzwa. Rakawedzera zvakanyanya kuyerera kweropa mumoyo (289.4% yakawedzera kuyerera kweropa mumoyo nebubble flowmeter) uye rakawedzera kuyerera kweropa muuropi neitsvo ne86.4% uye 64.5% paavhareji, izvo zvakasiyana zvakanyanya ne norepinephrine. Pakanga paine kudzikira kwekuyerera kweropa mumoyo uye kuwedzera kudiki asi kusingakoshi kwekushandiswa kweokisijeni mumoyo, izvo zvisina kuenderana nekuwedzera kukuru kwekuyerera kweropa mumoyo. Mukuedzwa kweECG mumbwa nenguruve yegaini, arrhythmia (ventricular tachycardia kana atrioventricular block) inokonzerwa nedosi yakawanda ye aurantii aurantii yakanga isiri yakakomba. Zvichibva pane zvataurwa pamusoro apa, zvakakurudzirwa kurapa cardiogenic shock. MaAlkaloids akaparadzaniswa kubva kuFructus Aurantii neLycium orange anogonawo kuwedzera kwenguva pfupi kushushikana kwetsandanyama dzakatsetseka dzeropa, kunyanya kana akarapwa nepituitrin.

4. Kudzivirira Kutapukira Kweropa: Kuongororwa kwemushonga weFructus Aurantii aqua decoction mu vitro kwakaratidza pachena kuti mushonga uyu unorwisa kutapukira kweropa.

5. Kurwisa allergy: 100mg/kg jekiseni remvura reFructus Aurantii Aurantii rinogona kudzivirira allergy yeganda (PCA) mumakonzo, uye 50μg/ml rinogona kudzivirira kuburitswa kwehistamine kubva mumasero emudumbu remakonzo.

6. Zvimwe zvinokonzerwa nazvo: Mycin yemuti weCitrus inogona kuderedza huwandu hwecholestatin muropa remakonzo anodyiswa chikafu chine cholesterol. Doro reFructus Aurantii rakaita kuti pave nemhedzisiro yekudzivirira mycobacterium tuberculosis H37Rv mu vitro, uye huwandu hwayo hwekudzivirira hwaive 1:1000. Muto wayo wemvura hauna kukanganisa paguinea pig bronchus. Zvakataurwa kuti muto wemichero yecitrus unowedzera mwero wekuvirisa uye hauderedzi kushanda kwawo mushure mekufashaira, saka hausi chikamu chema enzyme. Kushandiswa kukuru kwemuto weorenji mukurapa ndekwekuti wakapfuma muvhitamini C uye une huwandu hwakawanda hwevhitamini A neB. Peel haina vhitamini C asi yakapfuma muvhitamini A. Inonaka inovava uye inogona kusimbisa dumbu. Vana vakaita sekutora huwandu hwakawanda hwemapeel vanogona kukonzera chepfu (kurwadziwa kwemudumbu, kurwadziwa).

Chirevo: http://www.a-hospital.com

ZveCitrus Aurantium Extract, ndapota taurai nesu. Tiri kukumirirai pano chero nguva!!!

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Nguva yekutumira: Zvita-15-2022